Discover the new Chem-Impex: Where innovation starts with a bond.

Catalog Number:
17318
CAS Number:
290331-71-4
1-(tert-Butoxycarbonyl)-5-methoxy-1H-indol-2-ylboronic acid
Purity:
≥ 98% (HPLC)
Synonym(s):
1-Boc-5-methoxyindole-2-boronic acid
Documents
$40.00 /1G
Pack Size Availability Price
Request Bulk Quote
Product Information

1-(tert-Butoxycarbonyl)-5-methoxy-1H-indol-2-ylboronic acid is a versatile compound widely utilized in organic synthesis and medicinal chemistry. This boronic acid derivative is particularly valued for its ability to participate in Suzuki-Miyaura cross-coupling reactions, which are essential for forming carbon-carbon bonds in the development of complex organic molecules. Its unique structure, featuring a methoxy group and a tert-butoxycarbonyl protecting group, enhances its stability and reactivity, making it an ideal candidate for researchers looking to synthesize novel pharmaceuticals or advanced materials.

In addition to its synthetic applications, this compound has shown promise in the field of drug discovery, particularly in the development of targeted therapies. Its boronic acid functionality allows for the formation of reversible covalent bonds with diols, which is advantageous in designing inhibitors for various biological targets. Researchers and industry professionals can leverage the compound's properties to streamline their synthesis processes and enhance the efficacy of their drug candidates, ultimately contributing to advancements in therapeutic development.

Synonyms
1-Boc-5-methoxyindole-2-boronic acid
CAS Number
290331-71-4
Purity
≥ 98% (HPLC)
Molecular Formula
C14H18BNO5
Molecular Weight
291.11
MDL Number
MFCD04039006
PubChem ID
2794716
Melting Point
117 - 123 ?C
Appearance
Off-white powder
Conditions
Store at ≤ -4 °C
General Information
Synonyms
1-Boc-5-methoxyindole-2-boronic acid
CAS Number
290331-71-4
Purity
≥ 98% (HPLC)
Molecular Formula
C14H18BNO5
Molecular Weight
291.11
MDL Number
MFCD04039006
PubChem ID
2794716
Melting Point
117 - 123 ?C
Appearance
Off-white powder
Conditions
Store at ≤ -4 °C
Properties
Additional property information coming soon!
-
Safety and Regulations
Hazmat
No
Antibiotic
No
DEA-regulated
No
Warnings
-
Applications

1-(tert-Butoxycarbonyl)-5-methoxy-1H-indol-2-ylboronic acid is widely utilized in research focused on:

  • Pharmaceutical Development: This compound serves as a crucial intermediate in the synthesis of various pharmaceutical agents, particularly in the development of targeted cancer therapies.
  • Bioconjugation: It is employed in bioconjugation processes, allowing researchers to attach biomolecules to surfaces or other molecules, enhancing drug delivery systems.
  • Organic Synthesis: The compound is a valuable reagent in organic synthesis, facilitating the formation of complex molecules through cross-coupling reactions.
  • Material Science: It finds applications in the development of advanced materials, particularly in creating polymers with specific properties for electronics and coatings.
  • Analytical Chemistry: The compound is used in analytical methods for detecting and quantifying other substances, improving the accuracy of chemical analysis in various industries.

Citations