Discover the new Chem-Impex: Where innovation starts with a bond.

Catalog Number:
38022
CAS Number:
190791-29-8
Lasofoxifene tartrate
Purity:
≥ 98% (HPLC)
Synonym(s):
(5R,6S)-5,6,7,8-Tetrahydro-6-phenyl-5-[4-[2-(1-pyrrolidinyl)ethoxy]phenyl]-2-naphthalenol tartrate, Oporia
Documents
$111.17 /10MG
Pack Size Availability Price
Request Bulk Quote
Product Information

Lasofoxifene tartrate is a selective estrogen receptor modulator (SERM) that has garnered attention for its potential applications in women's health, particularly in the treatment and prevention of osteoporosis and breast cancer. This compound functions by selectively targeting estrogen receptors, offering a unique mechanism that can provide the benefits of estrogen without some of the associated risks. Researchers have noted its efficacy in improving bone density while minimizing the risk of endometrial hyperplasia, making it a promising alternative to traditional hormone replacement therapies.

In addition to its role in bone health, Lasofoxifene tartrate has shown potential in reducing the incidence of invasive breast cancer in postmenopausal women, positioning it as a valuable option in oncology. Its favorable pharmacological profile, including oral bioavailability and a manageable side effect profile, enhances its appeal for both clinical and research applications. As the demand for safer and more effective therapeutic agents continues to grow, Lasofoxifene tartrate stands out as a compound with significant potential in advancing women's health.

Synonyms
(5R,6S)-5,6,7,8-Tetrahydro-6-phenyl-5-[4-[2-(1-pyrrolidinyl)ethoxy]phenyl]-2-naphthalenol tartrate, Oporia
CAS Number
190791-29-8
Purity
≥ 98% (HPLC)
Molecular Formula
C28H31NO2·C4H6O6
Molecular Weight
563.65
MDL Number
MFCD30207839
PubChem ID
21706557
Melting Point
184 - 186 °C (dec.)
Appearance
White to almost white powder to crystal
Conditions
Store at 2 - 8 °C
General Information
Synonyms
(5R,6S)-5,6,7,8-Tetrahydro-6-phenyl-5-[4-[2-(1-pyrrolidinyl)ethoxy]phenyl]-2-naphthalenol tartrate, Oporia
CAS Number
190791-29-8
Purity
≥ 98% (HPLC)
Molecular Formula
C28H31NO2·C4H6O6
Molecular Weight
563.65
MDL Number
MFCD30207839
PubChem ID
21706557
Melting Point
184 - 186 °C (dec.)
Appearance
White to almost white powder to crystal
Conditions
Store at 2 - 8 °C
Properties
Additional property information coming soon!
-
Safety and Regulations
Hazmat
No
Antibiotic
No
DEA-regulated
No
Warnings
-
Applications

Lasofoxifene tartrate is widely utilized in research focused on:

  • Bone Health: This compound is studied for its potential to prevent osteoporosis by mimicking estrogen's beneficial effects on bone density, making it a valuable option for postmenopausal women.
  • Breast Cancer Treatment: Researchers are exploring its role as a selective estrogen receptor modulator (SERM) to inhibit the growth of estrogen-dependent breast tumors, providing a targeted approach in oncology.
  • Cardiovascular Health: Lasofoxifene tartrate is being investigated for its ability to positively influence lipid profiles, potentially reducing the risk of heart disease in women.
  • Menopausal Symptom Relief: The compound is evaluated for alleviating symptoms associated with menopause, such as hot flashes, offering a non-hormonal alternative to traditional hormone replacement therapies.
  • Research in Endocrinology: Its unique properties allow for studies on hormone receptor interactions, contributing to a deeper understanding of endocrine functions and disorders.

Citations